Naronapride - CAS 860174-12-5
Catalog number: 860174-12-5
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H41ClN4O5
Molecular Weight:
537.10
COA:
Inquire
Targets:
5-HT Receptor
Description:
Naronapride is a selective 5-HT(4) receptor agonist for gastrointestinal motility disorders. It can accelerate overall colonic transit and tend to accelerate GE and AC emptying and loose stool consistency. In Nov 2016, Renexxion planed two phase III trials for Constipation in USA.
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Purity:
98%
Appearance:
Powder
Synonyms:
860169-57-9(dihydrochloride); ATI7505; (R)-quinuclidin-3-yl 6-((3S,4R)-4-(4-amino-5-chloro-2-methoxybenzamido)-3-methoxypiperidin-1-yl)hexanoate
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Constipation
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
VGDDOIZXGFJDRC-VJTSUQJLSA-N
InChI:
InChI=1S/C27H41ClN4O5/c1-35-23-15-21(29)20(28)14-19(23)27(34)30-22-9-13-31(17-25(22)36-2)10-5-3-4-6-26(33)37-24-16-32-11-7-18(24)8-12-32/h14-15,18,22,24-25H,3-13,16-17,29H2,1-2H3,(H,30,34)/t22-,24+,25+/m1/s1
Canonical SMILES:
O=C(O[C@H]1CN2CCC1CC2)CCCCCN3C[C@H](OC)[C@H](NC(C4=CC(Cl)=C(N)C=C4OC)=O)CC3
Current Developer:
ARYx Therapeutics
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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