|Description||Nampt-IN-1, a pyridyloxyacetyl tetrahydroisoquinoline compound, is a novel inhibitor of nicotinamide phosphoribosyltransferase (NAMPT) with the potential to treat cancer. IC50: NCI-H1155 cell= 18 nM, Calu-6 cell= 49 nM, HCC1937 cell= 333 nM, MCF-7 cell= 3|
|Appearance||White to off-white Solid|
|Synonyms||2-hydroxy-2-methyl-N-[2-(2-pyridin-3-yloxyacetyl)-3,4-dihydro-1H-isoquinolin-6-yl]propane-1-sulfonamide Nampt-IN-1 CHEMBL3586462 SCHEMBL16634738|
|Solubility||DMSO: ≥ 45 mg/mL|
|Storage||Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -77℃ for long term (months to years).|
|Shelf Life||2 years|
|Boiling Point||659.9±65.0 °C | Condition: Press: 760 Torr|
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