Naltrindole hydrochloride - CAS 111469-81-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C26H27ClN2O3
Molecular Weight:
450.96
COA:
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Targets:
Opioid Receptor
Description:
Naltrindole hydrochloride is a cell permeable, potent and highly selective non-peptideδ opioid receptor antagonist (Ki= 0.02 nM) with 223- and 346-fold greater activity at δ than at μ and κ opioid receptors..
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Brife Description:
A highly potent and selective non-peptide δ opioid receptor antagonist (Ki= 0.02 nM)
Synonyms:
(4bS,8R,8aS,14bR)-7-(cyclopropylmethyl)-5,6,7,8,14,14b-hexahydro-4,8-methanobenzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol, monohydrochloride; Naltrindole (hydrochloride)
Solubility:
DMSO: ≥188 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
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InChIKey:
KNJKRQXCFJCQHC-UHFFFAOYSA-N
InChI:
1S/C26H26N2O3.ClH/c29-19-8-7-15-11-20-26(30)12-17-16-3-1-2-4-18(16)27-22(17)24-25(26,21(15)23(19)31-24)9-10-28(20)13-14-5-6-14;/h1-4,7-8,14,20,24,27,29-30H,5-6,9-13H2;1H
Canonical SMILES:
C1CC1CN2CCC34C5C6=C(CC3(C2CC7=C4C(=C(C=C7)O)O5)O)C8=CC=CC=C8N6.Cl
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Chemical Structure

CAS 111469-81-9 Naltrindole hydrochloride

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