MSC2530818 - CAS 1883423-59-3
Catalog number: B0084-007722
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C18H17ClN4O
Molecular Weight:
340.81
COA:
Inquire
Targets:
CDK
Description:
MSC2530818 is a specific and orally available CDK8 Inhibitor with an IC50 of 2.6 nM for CDK8.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-007722 10 mg $249 In stock
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Brife Description:
A specific and orally available CDK8 Inhibitor (CDK8 IC50 = 2.6 nM)
Synonyms:
MSC2530818; MSC-2530818; MSC 2530818. [(2S)-2-(4-chlorophenyl)pyrrolidin-1-yl]-(3-methyl-2H-pyrazolo[3,4-b]pyridin-5-yl)methanone; SCHEMBL17514257; s8387; AKOS032946259
Solubility:
DMSO: ≥125 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
576.5±50.0 ℃ at 760 Torr
Density:
1.373±0.06 g/cm3
InChIKey:
ODRITQGYYWHQGM-INIZCTEOSA-N
InChI:
1S/C18H17ClN4O/c1-11-15-9-13(10-20-17(15)22-21-11)18(24)23-8-2-3-16(23)12-4-6-14(19)7-5-12/h4-7,9-10,16H,2-3,8H2,1H3,(H,20,21,22)/t16-/m0/s1
Canonical SMILES:
CC1=C2C=C(C=NC2=NN1)C(=O)N3CCCC3C4=CC=C(C=C4)Cl
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CAS 1883423-59-3 MSC2530818

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