MRS 2365 - CAS 436847-09-5
Category: Inhibitor
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Molecular Formula:
C13H16N5O9P2SNa3
Molecular Weight:
549.28
COA:
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Targets:
P2Y Receptor
Description:
MRS 2365 is a highly potent, selective P2Y1 receptor agonist (EC50 = 0.4 nM), with no activity at P2Y12 receptors and only very low agonist activity at P2Y13 receptors (at concentrations up to 1 μM).
Purity:
≥98% by HPLC
Appearance:
Colourless liquid
Synonyms:
[[(1R,2R,3S,4R,5S)-4-[6-Amino-2-(methylthio)-9H-purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hex-1-yl]methyl] diphosphoric acid mono ester trisodium salt; MRS2365; MRS 2365; MRS-2365
Solubility:
Soluble in water (supplied pre-dissolved at a concentration of 10mM)
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
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InChIKey:
ZYPJOXVKTCEBCA-PVMCGCOJSA-K
InChI:
InChI=1S/C13H19N5O9P2S.3Na/c1-30-12-16-10(14)6-11(17-12)18(4-15-6)7-5-2-13(5,9(20)8(7)19)3-26-29(24,25)27-28(21,22)23;;;/h4-5,7-9,19-20H,2-3H2,1H3,(H,24,25)(H2,14,16,17)(H2,21,22,23);;;/q;3*+1/p-3/t5-,7?,8+,9+,13+;;;/m1.../s1
Canonical SMILES:
CSC1=NC2=C(C(=N1)N)N=CN2C3C4CC4(C(C3O)O)COP(=O)(O)OP(=O)(O)O
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Chemical Structure

CAS 436847-09-5 MRS 2365

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