|Description||MMV390048 is a novel antimalarial compound and it can competitively inhibit the binding of only a single protein, P. falciparum PI4 kinase, to the beads. MV390048 can become a child-friendly drug candidate for uncomplicated malaria that could be given as one single dose, completing the treatment in just one day. In May 2016, Phase I/II clinical trials in Malaria (In volunteers) in Australia was on-going.|
|Synonyms||UNII-0Z5T00JJ10;5-(4-(methylsulfonyl)phenyl)-6'-(trifluoromethyl)-[3,3'-bipyridin]-2-amine;MMV390048; MMV-390048; MMV 390048; MMV-048; MMV 048; MMV048.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Medicines for Malaria Venture; Technology Innovation Agency; University of Cape Town|
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