MLN1117 - CAS 1268454-23-4
Catalog number:
1268454-23-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H17N5O3
Molecular Weight:
363.37
COA:
Inquire
Targets:
PI3K
Description:
MLN1117, also known as INK1117, is a PI3Kα inhibitor which could lead to the apoptosis and growth retardation of tumor cells expressed by PI3Kα. IC50: 15 nM.
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Purity:
98%
Appearance:
Powder
Synonyms:
MLN1117; INK-1117; INK1117; [6-(2-amino-1,3-benzoxazol-5-yl)imidazo[1,2-a]pyridin-3-yl]-morpholin-4-ylmethanone;Serabelisib
Solubility:
DMSO: ≥ 6.4 mg/mL (Need ultrasonic or warming)
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
MLN1117 is a PI3Kα inhibitor which could lead to the apoptosis and growth retardation of tumor cells expressed by PI3Kα.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
BLGWHBSBBJNKJO-UHFFFAOYSA-N
InChI:
InChI=1S/C19H17N5O3/c20-19-22-14-9-12(1-3-16(14)27-19)13-2-4-17-21-10-15(24(17)11-13)18(25)23-5-7-26-8-6-23/h1-4,9-11H,5-8H2,(H2,20,22)
Canonical SMILES:
C1COCCN1C(=O)C2=CN=C3N2C=C(C=C3)C4=CC5=C(C=C4)OC(=N5)N
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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