ML281 - CAS 1404437-62-2
Catalog number: 1404437-62-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H19N3O2S
Molecular Weight:
389.47
COA:
Inquire
Targets:
Others
Description:
ML281, a quinoxalin derivative, has been found to be a STK33 inhibitor and could have probable effect against KRAS-dependent cancers. IC50: 14 nM.
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Purity:
98%
Appearance:
Powder
Synonyms:
ML281; CHEMBL2204239; Bg-stk33-59; MLS003876599; BRD8942; BRD-8942
Solubility:
5.6 μM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
ML281 has been found to be a STK33 inhibitor and could have probable effect against KRAS-dependent cancers.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Millgrams-Grams
InChIKey:
HWOYIOLMBQSTQS-UHFFFAOYSA-N
InChI:
InChI=1S/C22H19N3O2S/c1-13(2)14-9-10-16(24-21(26)19-8-5-11-28-19)15(12-14)20-22(27)25-18-7-4-3-6-17(18)23-20/h3-13H,1-2H3,(H,24,26)(H,25,27)
Canonical SMILES:
CC(C)C1=CC(=C(C=C1)NC(=O)C2=CC=CS2)C3=NC4=CC=CC=C4NC3=O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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