MK-2295 - CAS 878811-00-8
Catalog number: 878811-00-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H31FN6O2
Molecular Weight:
490.58
COA:
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Targets:
TRP Channel
Description:
MK-2295 is a potent TRPV1 antagonist. TRPV1 antagonists has the potential as analgesic and anti-inflammatory agents.
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Purity:
>98%
Appearance:
Solid powder
Synonyms:
6-[(3R)-4-[6-(4-fluorophenyl)-2-[(2R)-2-methylpyrrolidin-1-yl]pyrimidin-4-yl]-3-methylpiperazin-1-yl]-5-methylpyridine-3-carboxylic acid; 6-{4-[6-(4-Fluoro-phenyl)-2-(2-methyl-pyrrolidin-1-yl)-pyrimidin-4-yl]-3-(R)-methyl-piperazin-1-yl}-5-methyl-nicotinic acid; 3-​Pyridinecarboxylic acid, 6-​[(3R)​-​4-​[6-​(4-​fluorophenyl)​-​2-​[(2R)​-​2-​methyl-​1-​pyrrolidinyl]​-​4-​pyrimidinyl]​-​3-​methyl-​1-​piperazinyl]​-​5-​methyl-; 878811-00-8 (free base); 1855897-95-8 (mesylate salt)
MSDS:
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Canonical SMILES:
O=C(C1=CC(C)=C(N2C[C@@H](C)N(C3=NC(N4[C@H](C)CCC4)=NC(C5=CC=C(F)C=C5)=C3)CC2)N=C1)O
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