MK-0812 - CAS 624733-88-6
Catalog number: 624733-88-6
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C24H34F3N3O3
Molecular Weight:
469.54
COA:
Inquire
Targets:
CCR
Description:
Potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes
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Brife Description:
Potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes
Appearance:
Solid powder
Synonyms:
[(1S,3R)-3-[[(3S,4S)-3-methoxyoxan-4-yl]amino]-1-propan-2-ylcyclopentyl]-[3-(trifluoromethyl)-7,8-dihydro-5H-1,6-naphthyridin-6-yl]methanone
Solubility:
10 mM in DMSO
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS:
Inquire
Quality Standard:
In-house
Quantity:
Grams-Kilos
Boiling Point:
562oC at 760 mmHg
InChIKey:
MTMDXAIUENDNDL-RJSMDTJLSA-N
InChI:
1S/C24H34F3N3O3/c1-15(2)23(7-4-18(11-23)29-20-6-9-33-14-21(20)32-3)22(31)30-8-5-19-16(13-30)10-17(12-28-19)24(25,26)27/h10,12,15,18,20-21,29H,4-9,11,13-14H2,1-3H3/t18-,20+,21-,23+/m1/s1
Canonical SMILES:
CC(C)C1(CCC(C1)NC2CCOCC2OC)C(=O)N3CCC4=NC=C(C=C4C3)C(F)(F)F
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