Milveterol - CAS 652990-07-3
Catalog number:
652990-07-3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H29N3O4
Molecular Weight:
435.52
COA:
Inquire
Targets:
Adrenergic Receptor
Description:
Milveterol is a long-acting β(2)-adrenoceptor agonist. It is potentially useful for the treatment of chronic obstructive pulmonary disease (COPD) and asthma. It was developed by GlaxoSmithKline and Theravance together. It was in clinic phase 2 trials, but now it is terminated.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
GSK159797;N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[2-[4-[[(2R)-2-hydroxy-2-phenylethyl]amino]phenyl]ethylamino]ethyl]phenyl]formamide;GSK-159797
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Milveterol is potentially useful for the treatment of chronic obstructive pulmonary disease (COPD) and asthma.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
Boiling Point:
744.5±60.0 °C | Condition: Press: 760 Torr
Density:
1.307±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
BMKINZUHKYLSKI-DQEYMECFSA-N
InChI:
InChI=1S/C25H29N3O4/c29-17-28-22-14-20(8-11-23(22)30)24(31)15-26-13-12-18-6-9-21(10-7-18)27-16-25(32)19-4-2-1-3-5-19/h1-11,14,17,24-27,30-32H,12-13,15-16H2,(H,28,29)/t24-,25-/m0/s1
Canonical SMILES:
C1=CC=C(C=C1)C(CNC2=CC=C(C=C2)CCNCC(C3=CC(=C(C=C3)O)NC=O)O)O
Current Developer:
Milveterol was developed by GlaxoSmithKline and Theravance together. It was in clinic phase 2 trials, but now it is terminated.
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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