Mibefradil - CAS 116644-53-2
Catalog number:
116644-53-2
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C29H38FN3O3
Molecular Weight:
568.55
COA:
Inquire
Targets:
Calcium Channel
Description:
Mibefradil, a calcium channel blocker, has modest selectivity for T-type Ca2+ channels so that could be used in the treatment of sorts of cardiovascular disease like hypertension and chronic angina pectoris. IC50: 2.7 μM (for T-type).
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Purity:
>98 %
Appearance:
White solid
Synonyms:
Mibefradil;Mibefradil dihydrochloride
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
Mibefradil is a calcium channel blocker and has modest selectivity for T-type Ca2+ channels so that could be used in the treatment of sorts of cardiovascular disease like hypertension and chronic angina pectoris.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
HBNPJJILLOYFJU-VMPREFPWSA-N
InChI:
InChI=1S/C29H38FN3O3/c1-20(2)28-23-12-11-22(30)18-21(23)13-14-29(28,36-27(34)19-35-4)15-17-33(3)16-7-10-26-31-24-8-5-6-9-25(24)32-26/h5-6,8-9,11-12,18,20,28H,7,10,13-17,19H2,1-4H3,(H,31,32)/t28-,29-/m0/s1
Canonical SMILES:
CC(C)C1C2=C(CCC1(CCN(C)CCCC3=NC4=CC=CC=C4N3)OC(=O)COC)C=C(C=C2)F
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 116644-53-2 Mibefradil

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