MI-136 - CAS 1628316-74-4
Catalog number: 1628316-74-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H21F3N6S
Molecular Weight:
470.51
COA:
Inquire
Targets:
Androgen Receptor
Description:
MI-136, with the potential to treat refractory prostate cancer, inhibits DHT-induced expression of androgen receptor (AR) target genes. In vitro: Treatment with MI-136 inhibits the expression of genes that are bound to ASH2L after AR stimulation and induc
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Appearance:
Solid powder
Synonyms:
5-[[4-[[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino]piperidin-1-yl]methyl]-1H-indole-2-carbonitrile MI-136 5-((4-((6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl)amino)piperidin-1-yl)methyl)-1H-indole-2-carbonitrile 5-[(4-{[6-(2,2,2-Tri
Solubility:
DMSO: ≥ 31 mg/mL
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -39℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Grams-Kilos
Boiling Point:
654.9±55.0 °C | Condition: Press: 760 Torr
Density:
1.45±0.1 g/cm3
InChIKey:
PSOJDGBGVBEYJX-UHFFFAOYSA-N
InChI:
1S/C23H21F3N6S/c24-23(25,26)10-18-9-19-21(28-13-29-22(19)33-18)31-16-3-5-32(6-4-16)12-14-1-2-20-15(7-14)8-17(11-27)30-20/h1-2,7-9,13,16,30H,3-6,10,12H2,(H,28,29,31)
Canonical SMILES:
C1CN(CCC1NC2=C3C=C(SC3=NC=N2)CC(F)(F)F)CC4=CC5=C(C=C4)NC(=C5)C#N
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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