MGAT2-IN-1 - CAS 1800025-30-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H21ClF5N7O3S
Molecular Weight:
654.01
COA:
Inquire
Targets:
Others
Description:
An orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) (IC50= 7.8 for human, and 2.4 nM for mouse MGAT2).
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Synonyms:
N-(4-chloro-2,6-difluorophenyl)-1-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyrimidin-2-yl]-7-(2-oxopyrrolidin-1-yl)-2,3-dihydroindole-5-sulfonamide
Solubility:
DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
838.7±75.0 ℃ at 760 Torr
Density:
1.66±0.1 g/cm3
InChIKey:
VSZRYLHBOKTNBO-UHFFFAOYSA-N
InChI:
1S/C27H21ClF5N7O3S/c1-38-20(11-22(36-38)27(31,32)33)15-12-34-26(35-13-15)40-6-4-14-7-17(10-21(25(14)40)39-5-2-3-23(39)41)44(42,43)37-24-18(29)8-16(28)9-19(24)30/h7-13,37H,2-6H2,1H3
Canonical SMILES:
CN1C(=CC(=N1)C(F)(F)F)C2=CN=C(N=C2)N3CCC4=CC(=CC(=C43)N5CCCC5=O)S(=O)(=O)NC6=C(C=C(C=C6F)Cl)F
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 1800025-30-2 MGAT2-IN-1

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