|Description||Potent antagonist for α7-containing neuronal nicotinic receptors (Ki = 1.4 nM). Interacts with α4β2 and α6β2 receptors at concentrations > 40 nM. Attenuates METH-induced neurotoxicity in mouse striatum in vivo.|
|Purity||95 % (NMR).|
|Solubility||Slightly in methanol; not well in water, ethanol.|
|Storage||Store at +4 °C, in dark place;|
|Melting Point||185-187 °C.|
A substance which inhibits cholinesterases reversibly. Alkaloid , from plants of the Zygophyllaceae family
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Synthetic, a selective irreversible inhibitor of carboxylesterases
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