MDL 105519 - CAS 161230-88-2
Catalog number: 161230-88-2
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H11Cl2NO4
Molecular Weight:
376.19
COA:
Inquire
Targets:
NMDA Receptor
Description:
MDL 105519, a ligand selective for the glycine binding site of NMDA receptor, was shown that completely inhibited the binding of [3H]glycine to rat brain membranes with a Ki= 10.9±1.4 nM (n= 6). Inhibits [3H]glycine binding to the NMDA receptor with Kd= 3
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Appearance:
Solid powder
Synonyms:
3-[(E)-2-carboxy-2-phenylethenyl]-4,6-dichloro-1H-indole-2-carboxylic acid MDL 105,519 Mdl 105519 CHEMBL180427 (E)-4,6-Dichloro-3-(2-phenyl-2-carboxyethenyl)indole-2-carboxylic acid 161230-88-2 MDL-105519 Lopac-M-216 AC1O7G4O M216_SIGMA Lopac0_000805 C18H
Solubility:
DMSO:40 mg/mL
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -26℃ for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years
Quantity:
Grams-Kilos
Boiling Point:
601.3±55.0 °C | Condition: Press: 760 Torr
Density:
1.594±0.06 g/cm3
InChIKey:
LPWVUDLZUVBQGP-DHZHZOJOSA-N
InChI:
1S/C18H11Cl2NO4/c19-10-6-13(20)15-12(16(18(24)25)21-14(15)7-10)8-11(17(22)23)9-4-2-1-3-5-9/h1-8,21H,(H,22,23)(H,24,25)/b11-8+
Canonical SMILES:
C1=CC=C(C=C1)C(=CC2=C(NC3=CC(=CC(=C32)Cl)Cl)C(=O)O)C(=O)O
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