|Targets||CCR | HIV|
|Description||Selective CCR5 antagonist|
|B0084-067502||50 mg||$199||In stock|
|Brife Description||Selective CCR5 antagonist|
|Appearance||White to Off-White Solid|
|Synonyms||4,4-Difluoro-N-[(1S)-3-[(3-exo)-3-[3-methyl-5-(1-methylethyl-d6)-4H-1,2,4-triazol-4-yl]-8-azabicyclo[3.2.1]oct-8-yl]-1-phenylpropyl]cyclohexanecarboxamide; UK 427857-d6;|
|Solubility||Soluble to 75 mM in DMSO and to 100 mM in ethanol|
|Storage||Store at +4°C|
|Shelf Life||24 months.|
Potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes
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