LYC-55716 - CAS 2055536-64-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C27H23F6NO6S
Molecular Weight:
603.53
COA:
Inquire
Targets:
ROR
Description:
LYC-55716 is a first-in-class oral, small-molecule agonist of nuclear receptor retinoic acid–related orphan receptor γ (RORγ).
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Brife Description:
A novel oral RAR-related orphan receptor γ (RORγ) agonist
Synonyms:
3-[(2S)-6-[3-(difluoromethoxy)-5-fluorophenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2,2-dimethylpropanoic acid; SCHEMBL18302870
Solubility:
DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
669.1±65.0 ℃ at 760 Torr
Density:
1.417±0.06 g/cm3
InChIKey:
GULSIMHVQYBADX-FQEVSTJZSA-N
InChI:
1S/C27H23F6NO6S/c1-26(2,24(35)36)13-20-14-34(41(37,38)21-5-3-4-17(11-21)27(31,32)33)22-10-15(6-7-23(22)39-20)16-8-18(28)12-19(9-16)40-25(29)30/h3-12,20,25H,13-14H2,1-2H3,(H,35,36)/t20-/m0/s1
Canonical SMILES:
CC(C)(CC1CN(C2=C(O1)C=CC(=C2)C3=CC(=CC(=C3)F)OC(F)F)S(=O)(=O)C4=CC=CC(=C4)C(F)(F)F)C(=O)O
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CAS 2055536-64-4 LYC-55716

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