LY3009120 - CAS 1454682-72-4
Catalog number:
1454682-72-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H29FN6O
Molecular Weight:
424.51
COA:
Inquire
Targets:
Raf
Description:
LY03009120 is a potent pan-Raf inhibitor with IC50 of 44 nM, 31-47 nM, and 42 nM for A-raf, B-Raf, and C-Raf in A375 cells, respectively. Phase 1.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
LY-3009120; LY 3009120; DP4978; DP 4978; DP-4978.
Solubility:
DMSO,3mg/mLwarmed(7.06mM);Water,<1mg/mL(<1mM);Ethanol,<1mg/mLwarmed(<1mM)
Storage:
3 years -20℃powder;6 months-80℃in solvent
MSDS:
Inquire
Shelf Life:
2 years if stored properly
Canonical SMILES:
O=C(NC1=CC(C2=CC3=CN=C(NC)N=C3N=C2C)=C(C)C=C1F)NCCC(C)(C)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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