LY2606368 dihydrochloride - CAS 1234015-54-3
Catalog number:
1234015-54-3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H21Cl2N7O2
Molecular Weight:
438.31
COA:
Inquire
Targets:
Checkpoint Kinase (Chk)
Description:
The dihydrochloride salt form of LY2606368 which also known as prexasertib, is an inhibitor of checkpoint kinase 1 and has potential effect in antineoplastic. It is still under Phase II clinical trial against breast cancer and some other sorts of cancers.
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Purity:
98%
Appearance:
Powder
Synonyms:
UNII-9RFT476U2L; 9RFT476U2L; LY2606368 (dihydrochloride); 1234015-54-3; HY-18174A; CS-3507
Solubility:
43mg/ml in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
The dihydrochloride salt form of LY2606368 which also known as prexasertib, is an inhibitor of checkpoint kinase 1 and has potential effect in antineoplastic.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
KMEIPKXRCJTZBZ-UHFFFAOYSA-N
InChI:
InChI=1S/C18H19N7O2.2ClH/c1-26-14-4-2-5-15(27-7-3-6-19)18(14)13-8-16(25-24-13)23-17-11-21-12(9-20)10-22-17;;/h2,4-5,8,10-11H,3,6-7,19H2,1H3,(H2,22,23,24,25);2*1H
Canonical SMILES:
COC1=C(C(=CC=C1)OCCCN)C2=CC(=NN2)NC3=NC=C(N=C3)C#N.Cl.Cl
Current Developer:
Eli Lilly/National Cancer Institute (USA)
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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