|Description||LY-79771 is a antiobesity agent. It can be effective in preventing fat regain following energy deprivation.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
GYKI-23107 is an antiarrhythmic agent with local anaesthetic activity.
Cot inhibitor-2 is a COT/Tpl2 inhibitor.
Gemcabene is an orally available lipid-lowering small molecule designed to target known lipid metabolic pathways, as an adjunctive therapy to reduce LDL-C, hsCR...
This active molecular is a selective peptide deformylase inhibitor. It has good anti-bacteria activity in vitro. Antibacterial spectrum of Lanopepden includes S...
Amfebutamone (Bupropion) HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrin...
Indirubin is an inhibitor of GSK-3β and of cyclin-dependent kinases (CDK1/cyclin B, CDK2/cyclin A, CDK2/cyclin E, CDK4/cyclin D1, CDK5/p35). Also, indirubin is ...
3PO is originally reported to inhibit PFKFB3 (IC50 = 25 μM), with the potential to inhibit cancer cell proliferation. The addition of selective inhibitors of au...
Icariin is a flavonol glycoside, a type of flavonoid. Icariin is a PDE5 inhibitor with IC50 of 0.432 μM, 167-fold more selective for PDE5 than PDE4.
Coptisine chloride, an alkaloid found in Chinese goldthread, can be absorbed across intestinal epithelial cells, and they are completely absorbed compounds.
Carbazochrome sodium sulfonate (AC-17)
Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for use in the treatment of hemorrhoids.
Mecarbinate is a chemical intermediate of arbidol hydrochloride.
TC-O9311 is a potent, selective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139) with no activity against a range of 90 diverse targets.
Tafamidis is a potent and selective transthyretin kinetic stabilizer that inhibits the amyloid cascade. It is a drug for the amelioration of transthyretin-relat...
Tetracaine is a topical local anesthetic for the eyes. It works by interfering with entry of sodium ions into nerve cells. It is also used in assessing the pote...
Sodium Nitroprusside is a potent vasodilator working through releasing NO spontaneously in blood.
Cgp 43902A is a bio-active molecular, but no detailed information has been published yet.
Thiamet G is a potent, selective O-GlcNAcase inhibitor with Kiof 21 nM, while exhibiting 37,000-fold selectivity over human lysosomal –hexosaminidase.
KPU-300, a diketopiperazine derivative, has been found to be an antimicrotubule agent and exhibit cytotoxicity against HT-29 cells. IC50: 7.0 nM.
Clonidine is an α2-Adrenergic agonist for neuropathic pain.