LY-411575 isomer 3
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C26H23F2N3O4
Molecular Weight:
479.48
COA:
Inquire
Targets:
γ-secretase
Description:
LY-411575 isomer 3, is an isomer of LY411575, which is a potent, cell-permeable γ-secretase inhibitor (IC50= 0.078 nM/0.082 nM (in membrane-assay/in cell-basedγ-secretase assays)) and also inhibits Notch clevage (IC50= 0.41 nM). Phase III
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Brife Description:
Inhibits γ-secretase and Notch clevage
Appearance:
White to off-white solid
Synonyms:
LY411575 isomer 3; LY 411575 isomer 3
Solubility:
Soluble to 98 mg/mL in DMSO
Storage:
Store in a cool and dry place and at 0 - 4℃ for short term (days to weeks) or -41℃ for long term (months to years).
MSDS:
Inquire
Boiling Point:
836.0±65.0℃ at 762 Torr
Density:
1.40±0.1 g/cm5
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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