LY 106737 - CAS 82970-72-7
Catalog number: 82970-72-7
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21-H27-N-O
Molecular Weight:
309.45
COA:
Inquire
Targets:
Opioid Receptor
Description:
LY 106737 is phenylpiperidine opioid receptor antagonist, but no detailed information has been published yet.
Publictions citing BOC Sciences Products
  • >> More
Purity:
98%
Appearance:
Powder
Synonyms:
cis-(+-)-3-(3,4-dimethyl-1-(2-phenylethyl)-4-piperidinyl)-Phenol
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
ULOGPOOAAOSAOC-LAUBAEHRSA-N
InChI:
1S/C21H27NO/c1-17-16-22(13-11-18-7-4-3-5-8-18)14-12-21(17,2)19-9-6-10-20(23)15-19/h3-10,15,17,23H,11-14,16H2,1-2H3/t17-,21+/m0/s1
Canonical SMILES:
C[C@H]1CN(CC[C@@]1(C)c2cccc(c2)O)CCc3ccccc3
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Opioid Receptor Products


CAS 152657-84-6 Nalfurafine

Nalfurafine
(CAS: 152657-84-6)

Nalfurafine is a selective and centrally-penetrant κ-opioid receptor (KOR) agonist without significant activity on μ- and δ-opioid receptors. With antipruritic ...

CAS 58-74-2 Papaverine

Papaverine
(CAS: 58-74-2)

Papaverine is an opiate alkaloid isolated from the plant Papaver somniferum. It is used primarily in the treatment of visceral spasm, vasospasm. It is also used...

CAS 825649-28-3 JNJ 20788560

JNJ 20788560
(CAS: 825649-28-3)

JNJ-20788560 is a delta opioid agonist analgesics. No recent reports of development identified for preclinical development in Inflammatory-pain in USA.

CAS 59263-76-2 Meptazinol Hydrochloride

Meptazinol Hydrochloride
(CAS: 59263-76-2)

Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]-dihydromorphine binding with IC50 of 58 nM.

CAS 133267-27-3 Fedotozine tartrate

Fedotozine tartrate
(CAS: 133267-27-3)

Fedotozine tartrate is a kappa(1a) opioid receptor agonist.

CAS 1401031-39-7 TRV130 HCl

TRV130 HCl
(CAS: 1401031-39-7)

TRV130 is an opioid drug that is under evaluation in human clinical trials for the treatment of acute severe pain. It is a functionally selective μ-opioid recep...

Alvimopan monohydrate
(CAS: 1383577-62-5)

The monohydrate salt form of Alvimopan could be commonly used in postoperative recovery of gastrointestinal for acting as a mu-opioid receptor (PAM-OR) antagoni...

CAS 1108147-88-1 MCOPPB triHydrochloride

MCOPPB triHydrochloride
(CAS: 1108147-88-1)

The trihydrochloride salt form of MCOPPB, an effective full agonist of nociceptin receptor, could be a good antianxiety agent with few side-effects. pKi: 10.07.

CAS 244218-51-7 JTC-801

JTC-801
(CAS: 244218-51-7)

JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ. It is an opioid analgesic dru...

CHIR 4531
(CAS: 158198-48-2)

CHIR 4531, an oligopeptides compound, has been found to be an opioid mu receptor agonist and was once studied in pain therapy.

CAS 189388-22-5 Endomorphin 1

Endomorphin 1
(CAS: 189388-22-5)

Endomorphin 1 is a high affinity (Ki = 360 pM) and highly selective agonist of theμ-opioid receptor with 4000- and 15000-fold preference over δ and κ respective...

CAS 850173-95-4 ADL5859 HCl

ADL5859 HCl
(CAS: 850173-95-4)

ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel.

CAS 785835-79-2 JDTic dihydrochloride

JDTic dihydrochloride
(CAS: 785835-79-2)

JDTic dihydrochloride is a highly selective antagonist for the κ-opioid receptor with IC50 value of 0.02nM without affecting the μ- or δ-opioid receptors. It is...

LY2795050
(CAS: 1346133-08-1)

LY2795050, a κ-opioid Receptor antagonist, has been found to be effective in imaging KOR behaving as a PET tracer. IC50: 0.72 nM and 25.8 nM for κ-opioid Recept...

LY 106737
(CAS: 82970-72-7)

LY 106737 is phenylpiperidine opioid receptor antagonist, but no detailed information has been published yet.

TRV130
(CAS: 1401028-24-7)

TRV130 is an oxaspiro compound that has been found to be a μ-opioid receptor G protein ligand and could be used in pain therapy. IC50: 8.1 (pEC50. G protein ass...

CAS 34140-59-5 Trimebutine Maleate

Trimebutine Maleate
(CAS: 34140-59-5)

Trimebutine is an opioid receptor agonist used as spasmolytic agent abdominal pain.

CAS 58569-55-4 Met-Enkephalin

Met-Enkephalin
(CAS: 58569-55-4)

Met-Enkephalin is synthetic opioid peptides that has opioid effects of a relatively short duration.

CAS 111469-81-9 Naltrindole hydrochloride

Naltrindole hydrochloride
(CAS: 111469-81-9)

Naltrindole hydrochloride is a cell permeable, potent and highly selective non-peptideδ opioid receptor antagonist (Ki= 0.02 nM) with 223- and 346-fold greater ...

GSK1521498
(CAS: 1007573-18-3)

GSK-1521498 is a novel μ-Opioid receptor antagonist. It shows to attenuate reward-driven compulsive behaviours, such as stimulant drug seeking or binge eating i...

Quick Inquiry

Verification code

Featured Items