|Description||Lusaperidone, also known as R107474, is an α2 adrenergic receptor antagonist. R107474 showed high affinity for ha2A-, ha2B-, and ha2C-adrenoceptors, stably expressed in CHO cells. The compound bound preferentially to the ha2A- and ha2C-adrenoceptor subtypes (Ki = 0.13 and 0.15 nM, respectively) and was seven times less potent in binding to the ha2B-adrenoceptors (Ki = 1.03 nM).|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||538.3±60.0 ℃ at 760 Torr|
Guanabenz Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respe...
Spiroxatrine is a 5-HT1A antagonist and a potent α2C adrenergic receptor antagonist. Spiroxatrine exhibits great anxiolytic effects in combination with buspiron...
The hydrochloride of Nifenalol. Nifenalol is a beta-adrenoceptor antagonist used for the treatment of cardiovascular and cerebrovascular diseases such as hypert...
Tolazoline is a non-selective competitive α-adrenergic receptor antagonist.
Terbutaline, also called as Bronclyn, as a fast-acting bronchodilator it is a β2 adrenergic receptor agonist used to treat asthma and premature labor.
Efaroxan hydrochloride is a potent and selective α2 adrenoceptor antagonist and imidazoline I1 receptor ligand (pKi = 7.87, 7.42, 5.74, 7.28 and < 5 for α 2A, α...
Oxymetazoline, an imidazol derivative, has been found to be an adrenergic receptor agonist that could be an effective topical decongestant.
Isoetarine is a selective adrenergic beta-2 agonist. It is used as fast acting bronchodilator for emphysema, bronchitis and asthma. It has been listed.
Xamoterol hemifumarate is a third generation β1-adrenoceptor-selective partial agonist (pA2 = 7.4 - 7.8 and 5.2 - 6.2 at β1- and β2-adrenoceptors, respectively)...
Pronethalol is a non-selective beta-adrenergic blocking agentused in treatment due to carcinogenic properties.
MK-351 hydrochloride is an alpha-adrenergic agonist selective for α2-adrenergic receptors. It is a psychoactive drug used as a sympatholytic or antihypertensive...
Brombuterol is found to be a novel β-adrenergic agonist that can increase the meat-to-fat ratio but it is banned in animal feeds.
Propranolol hydrochloride, with antihypertensive, antianginal and antiarrhythmic (class II) properties, is a non-cardioselective adrenergic-beta antagonist and ...
Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn..
Esmolol is a cardioselective beta1 receptor blocker with rapid onset, a very short duration of action, and no significant intrinsic sympathomimetic or membrane ...
AH 11110 hydrochloride
The hydrochloride salt form of AH 11110, which is an α1B-adrenoceptor ligand and has been found to exhibit interaction with α1-adrenoceptors as well as α2-adren...
Clorprenaline is a beta-adrenergic receptor agonist.
BRL 44408 maleate
BRL 44408 maleate is a selective α2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at α2A and α2B-adrenergic receptors, respectively). BRL 44408 increases h...
Levobunolol hydrochloride, a beta1- and beta2-adregergic blocking agent, has proved to be an effective ocular hypotensive agent to treat glaucoma.
The mesylate salt form of Dihydroergotamine, which has been found to be a partial α-adrenergic agonist and could be used as an antimigraine agent.