Lu AE58054 - CAS 467459-31-0
Catalog number:
467459-31-0
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20H19F5N2O
Molecular Weight:
398.37
COA:
Inquire
Targets:
5-HT Receptor
Description:
Lu AE58054 is a selective and high affinity 5-HT6 receptor antagonist as promising treatment for cognitive disorders.
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Purity:
≥98%
Related CAS:
467458-02-2 (HCl salt)
Appearance:
Solid powder
Synonyms:
2-(6-fluoro-1H-indol-3-yl)-N-(3-(2,2,3,3-tetrafluoropropoxy)benzyl)ethanamine; Lu AE58054; Lu AE-58054; Lu AE 58054; Idalopirdine; Iladopirdine
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
5-HT(6)R antagonist
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
YBAWYTYNMZWMMJ-UHFFFAOYSA-N
InChI:
1S/C20H19F5N2O/c21-15-4-5-17-14(11-27-18(17)9-15)6-7-26-10-13-2-1-3-16(8-13)28-12-20(24,25)19(22)23/h1-5,8-9,11,19,26-27H,6-7,10,12H2
Canonical SMILES:
FC1=CC2=C(C=C1)C(CCNCC3=CC=CC(OCC(F)(F)C(F)F)=C3)=CN2
Current Developer:
Lundbeck A/S; Otsuka Pharmaceutical
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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