|Description||LPA2 antagonist 1 could block the Erk activation regulated by LPA(2) and proliferation of HCT-116 cells as a selective inhibitor of LPA2 protein. IC50: 17 nM (in vitro). It could also be used to assess the inhibiting effection in the process of anticancer|
|Synonyms||LPA2 antagonist 1; CHEMBL256470; BDBM50373826; AKOS027314118; CS-3103; AK298931|
|Solubility||10 mM in DMSO|
|Application||LPA2 antagonist 1 could block the Erk activation regulated by LPA(2) and proliferation of HCT-116 cells as a selective inhibitor of LPA2 protein.|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly|
LPA2 antagonist 1
LPA2 antagonist 1 could block the Erk activation regulated by LPA(2) and proliferation of HCT-116 cells as a selective inhibitor of LPA2 protein. IC50: 17 nM (i...
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