LPA2 antagonist 1 - CAS 1017606-66-4
Catalog number:
1017606-66-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20H23Cl2N5O2S2
Molecular Weight:
500.46
COA:
Inquire
Targets:
LPL Receptor
Description:
LPA2 antagonist 1 could block the Erk activation regulated by LPA(2) and proliferation of HCT-116 cells as a selective inhibitor of LPA2 protein. IC50: 17 nM (in vitro). It could also be used to assess the inhibiting effection in the process of anticancer
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Purity:
95%
Appearance:
Powder
Synonyms:
LPA2 antagonist 1; CHEMBL256470; BDBM50373826; AKOS027314118; CS-3103; AK298931
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
LPA2 antagonist 1 could block the Erk activation regulated by LPA(2) and proliferation of HCT-116 cells as a selective inhibitor of LPA2 protein.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
BPRNMVDTWIHULJ-AWEZNQCLSA-N
InChI:
InChI=1S/C20H23Cl2N5O2S2/c1-13-11-30-19-18(13)23-12-24-20(19)25-14(2)10-26-5-7-27(8-6-26)31(28,29)15-3-4-16(21)17(22)9-15/h3-4,9,11-12,14H,5-8,10H2,1-2H3,(H,23,24,25)/t14-/m0/s1
Canonical SMILES:
CC1=CSC2=C1N=CN=C2NC(C)CN3CCN(CC3)S(=O)(=O)C4=CC(=C(C=C4)Cl)Cl
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