Lisuride maleate - CAS 19875-60-6
Catalog number: 19875-60-6
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H31N3O5
Molecular Weight:
454.58
COA:
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Targets:
Dopamine Receptor
Description:
Lisuride maleate, an ergot derivative, is a nonselective dopamine receptor agonist with high affinity for D2, D3 and D4 receptors along with 5-HT1A. As an anti-Parkinson's agent with anticonvulsive effects, Lisuride maleate has been shown to decrease the release of prolactin and reduce inflammatory mediators such as IL6 and TNF-α.
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Purity:
>99 %
Appearance:
White Solid
Synonyms:
3-[(6aR,9S)-7-methyl-6,6a,8,9-tetrahydro-4H-indolo[4,3-fg]quinoline-9-yl]-1,1-diethylurea;(Z)-but-2-enedioic acid; Lisuride Maleate ; Cuvalit; Lysenyl; Lysenyl bimaleate; Lysenyl hydrogen maleate; Lisuride hydrogen maleate; Mesylate, Lisuride; Methylergol ;Carbamide Revanil
MSDS:
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Boiling Point:
836.3℃ at 760 mmHg
InChIKey:
CVQFAMQDTWVJSV-BAXNFHPCSA-N
InChI:
1S/C20H26N4O.C4H4O4/c1-4-24(5-2)20(25)22-14-10-16-15-7-6-8-17-19(15)13(11-21-17)9-18(16)23(3)12-14;5-3(6)1-2-4(7)8/h6-8,10-11,14,18,21H,4-5,9,12H2,1-3H3,(H,22,25);1-2H,(H,5,6)(H,7,8)/b;2-1-/t14-,18+;/m0./s1
Canonical SMILES:
CCN(CC)C(=O)NC1CN(C2CC3=CNC4=CC=CC(=C34)C2=C1)C.C(=CC(=O)O)C(=O)O
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Chemical Structure

CAS 19875-60-6 Lisuride maleate

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