|Description||Lidocaine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.|
QS11 contains a planar purine ring with C2, C6, and N9-positions substituted. QS11, a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor...
FMK 9a is a covalent autophagin-1 inhibitor (IC50= 80 and 73 μM in FRET and LRA assay).
An alkaloid FR 5 from Fritillaria thunbergii. An angiotensin converting enzyme inhibitory steroidal alkaloid. It is a commonly used antitussive and expectorant ...
Rhynchophylline and isorhynchophylline act as noncompetitive antagonists of the NMDA receptor and that this property may contribute to the neuroprotective and a...
BVT 2733 is a non-steroidal small molecule as a a selective 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor (IC = 96 ± 14 nM w).
TAK-683 is an investigational peptide derivative of metastin under the development of Millennium. It is a KISS1R protein agonist. Phase I development for prosta...
Albiflorin is a major constituent presents in peony root, which possesses therapeutic potential for neurodegenerative diseases.
CS-M1996 is a 4′-Azidocytidine analogue. It can inhibit Hepatitis C virus replication.
BMS 182264 is a bio-active chemical, but few detailed information has been published yet.
Sodium Danshensu is a mono sodium of danshensu, which is a natural phenolic acid of caffeic acid derivatives isolated from Salvia miltiorrhiza.
Benserazide HCl is a peripherally-acting aromatic L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.
Ginsenoside Rc, a sort of triterpene saponin, is extracted from ginseng and has been found to be antioxidative, anti-aging and has sorts of other properties. It...
Difluprednate (difluoroprednisolone butyrate acetate, or DFBA) is a synthetic difluorinated prednisolone derivative, it is originally developed for dermatologic...
Prostanoid GD(2) is released from mast cells in response to allergen challenge. AM156 is a selective prostanoid DP(2) receptor antagonist and it inhibits sneezi...
LY 186564 is a bio-active chemical,but no detailed information has been published yet.
Extract from the roots of Coptis chinensis Franch, shows strong activity with IC50 48.1 µM.
Phenformin HCl is a hydrochloride salt of phenformin that is an anti-diabetic drug from the biguanide class.
Ginsenoside Rf, extracted from the traditional Chinese herb ginseng used as an aldose reductase inhibitor and exert anti-inflammatory and immunomodulatory activ...
Mas7, a structural analogue of mastoparan, is G protein activator via Gαi and Gαo stimulation.