LH846 - CAS 639052-78-1
Catalog number: B0084-463302
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C16H13ClN2OS
Molecular Weight:
316.81
COA:
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Targets:
CK1
Description:
LH846 is a selective inhibitor of CK1δ, which displays no inhibitory activity at CK2. It inhibits CK1δ-dependent phosphorylation and degradation of PER1 protein, showing to lengthen the circadian period in U2OS cells, with minimal effect on amplitude.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-463302 50 mg $248 In stock
B0084-463302 100 mg $448 In stock
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Purity:
>98%
MSDS:
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InChIKey:
DYHAMRNAHTWYKY-UHFFFAOYSA-N
InChI:
InChI=1S/C16H13ClN2OS/c1-10-7-14-13(9-12(10)17)18-16(21-14)19-15(20)8-11-5-3-2-4-6-11/h2-7,9H,8H2,1H3,(H,18,19,20)
Canonical SMILES:
CC1=CC2=C(C=C1Cl)N=C(S2)NC(=O)CC3=CC=CC=C3
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CAS 639052-78-1 LH846

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