LGD-6972 - CAS 1207989-09-0
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C43H46N2O5S
Molecular Weight:
702.9
COA:
Inquire
Targets:
Glucagon Receptor
Description:
LGD-6972 is an orally bioavailable small molecule glucagon receptor antagonist being developed as an adjunct to diet and exercise to improve glycemic control in adults with T2DM.
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Brife Description:
A glucagon receptor antagonist
Synonyms:
2-[[4-[(2R)-2-[4-(4-tert-butylphenyl)phenyl]-3-oxo-3-[4-(2,4,6-trimethylphenyl)anilino]propyl]benzoyl]amino]ethanesulfonic acid
Solubility:
DMSO: ≥ 31 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Density:
1.206±0.06 g/cm3
InChIKey:
HKJMCBYPVCGZFB-LDLOPFEMSA-N
InChI:
1S/C43H46N2O5S/c1-28-25-29(2)40(30(3)26-28)35-17-21-38(22-18-35)45-42(47)39(27-31-7-9-36(10-8-31)41(46)44-23-24-51(48,49)50)34-13-11-32(12-14-34)33-15-19-37(20-16-33)43(4,5)6/h7-22,25-26,39H,23-24,27H2,1-6H3,(H,44,46)(H,45,47)(H,48,49,50)/t39-/m1/s1
Canonical SMILES:
CC1=CC(=C(C(=C1)C)C2=CC=C(C=C2)NC(=O)C(CC3=CC=C(C=C3)C(=O)NCCS(=O)(=O)O)C4=CC=C(C=C4)C5=CC=C(C=C5)C(C)(C)C)C
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CAS 1207989-09-0 LGD-6972

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