Lexibulin - CAS 917111-44-5
Catalog number:
917111-44-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
COA:
Inquire
Targets:
Microtubule/Tubulin
Description:
lexibulin, also known as CYT997,  is an orally bioavailable small-molecule with tubulin-inhibiting, vascular-disrupting, and potential antineoplastic activities. Lexibulin inhibits tubulin polymerization in tumor blood vessel endothelial cells and tumor cells, blocking the formation of the mitotic spindle and leading to cell cycle arrest at the G2/M phase; this may result in disruption of the tumor vasculature and tumor blood flow, and tumor cell death. Check for active clinical trials or closed clinical trials using this agent. (NCI Thesaurus)
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Appearance:
white solid powder
Synonyms:
CYT997; CYT-997; CYT 997. lexibulin.
MSDS:
Inquire
Current Developer:
YM BioSciences Australia Pty Ltd.
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CAS 917111-44-5 Lexibulin

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