Lexanopadol - CAS 1357348-09-4
Catalog number:
1357348-09-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H25FN2O
Molecular Weight:
364.46
COA:
Inquire
Targets:
Opioid Receptor
Description:
Lexanopadol is a potent Opioid mu receptor agonist originated by Grunenthal. Lexanopadol is suited for the management of moderate to severe chronic pain, including neuropathic pain. No recent reports of development were identified for phase-I development in Pain in Germany
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Purity:
98%
Appearance:
Powder
Synonyms:
(1r,4r)-6'-fluoro-N-methyl-4-phenyl-4',9'-dihydro-3'H-spiro[cyclohexane-1,1'-pyrano[3,4-b]indol]-4-amine;trans-6'-Fluoro-N-methyl-4-phenyl-4',9'-dihydro-3'H-spiro(cyclohexane-1,1'-pyrano(3,4-b)indol)-4-amine;GRT6006
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Pain
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
AMXGKMSRYLZAEO-YHBQERECSA-N
InChI:
1S/C23H25FN2O/c1-25-22(16-5-3-2-4-6-16)10-12-23(13-11-22)21-18(9-14-27-23)19-15-17(24)7-8-20(19)26-21/h2-8,15,25-26H,9-14H2,1H3/t22-,23-
Canonical SMILES:
CN[C@]1(CC[C@]2(OCCc3c2[nH]c4c3cc(cc4)F)CC1)c5ccccc5
Current Developer:
Originator Grunenthal
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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