|Description||Levonordefrin is a adrenergic receptor agonist and can be used as a topical nasal decongestant and vasoconstrictor in dentistry in the United States. Levonordefrin is also a metabolite of the antihypertensive drug methyldopa.|
|Appearance||White to Pale Beige Solid|
|Synonyms||4-[(1R,2S)-2-Amino-1-hydroxypropyl]-1,2-benzenediol; BA 2818; Corbadrine; D-(-)-Cobefrin; L-α-Methylnoradrenaline; Levonordefrin; Neo-cobefrin; l-Cobefrin; (-)-Nordefrin;|
|Solubility||Acidic Aqueous, DMSO (Sparingly)|
|Shelf Life||2 month in rt, long time|
|Boiling Point||No Data Available|
|Melting Point||>200℃ (dec.)|
Carmoterol, a quinolin derivative, has been found to a β2-adrenoceptor agonist that could be an effective bronchodilating agent.
Metoprolol is a a selective β1 receptor blocker for the treatment of a variety of cardiovascular disorder.
SNAP 5089 is an α1A-adrenoceptor antagonist with > 600-fold selectivity over other adrenoceptors (Ki = 0.35, 220, 370, 540, 800 and 1200 nM for α1A, α1B, α2C, α...
Cimbuterol is a β-adrenergic agonist.
Bisoprolol is a beta-adrenoceptor blocking drug (beta-blocker). More specifically, it is a selective type β1 adrenergic receptor blocker.
MK-0634, also called as L-796568, is an β3 adrenergic receptor agonist that was progressed into clinical studies for the treatment of obesity in the early 2000s...
ABT-866 is a novel alpha-adrenoceptor agent that demonstrates intrinsic activity at the α1A-adrenoceptor subtype present in the rabbit urethra (pD2=6.22, with 8...
This active molecular is a β-adrenergic receptor antagonist. Levonebivolol is an enantiomer of Nebivolol which is a β1 receptor blocker with nitric oxide-potent...
Naftopidil hydrochloride is an α1-adrenoceptor antagonist with only weak antagonism at post-junctional α2 receptors. Used as a potent, persistent antihypertensi...
Scopine is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
Carvedilol phosphate hemihydrate is a nonselective beta (β1, β2) blocker and alpha (α1) blocker, inhibits LDL oxidation (IC50 = 3.8 μM).
Guanfacine Hydrochloride is a centrally acting alpha-2 adrenergic agonist that has been available as an FDA-approved hypotensive agent for more than two decades...
Salmefamol is a beta2-adrenoceptor agonist which is useful for treatment of respiratory diseases.
ICI 89406 is a selective β-adrenergic antagonist. It is a low efficacy partial agonist and does not affect resting cardiac parameters.
CGP-12388 is a beta-adrenoceptor antagonist-derived radioligands. It is used for cardiac PET imaging due to its high hydrophilicity and affinity to beta-adrenoc...
Lerimazoline is an α-adrenergic receptor agonist. It inhibits secretion of nasal mucus. It causes hypertension. It is common used in the form of hydrochloride.
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstru...
Guanadrel, as an antihypertensive agent, is an orally active postganglionic sympathetic inhibitor.
An S enantiomer which has affinity at alpha 1 adrenergic receptor
Naphazoline is Alpha adrenergic receptor agonist. It is a vasoconstrictor with a rapid action in reducing swelling when applied to mucous membrane. It acts on a...