|Description||Levocabastine is a selective second-generation Histamine H1 receptor antagonist. It is used for Allergic conjunctivitis and Seasonal allergic rhinitis。Levocabastine is also a potent and selective antagonist for the neurotensin receptor NTS2 and it can be used to characterise the different neurotensin subtypes.|
|Synonyms||Levocabastine, Livostin, Bilina;(3S,4R)-1-[4-cyano-4-(4-fluorophenyl)cyclohexyl]-3-methyl-4-phenylpiperidine-4-carboxylic acid|
|Solubility||Soluble in DMSO|
|Application||Allergic conjunctivitis; Seasonal allergic rhinitis|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Janssen-Cilag; Kyowa Hakko Kirin; Nippon Shinyaku; Santen Pharmaceutical|
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