|Description||LB-100 is a water solubleprotein phosphatase 2A (PP2A)inhibitor(IC50= 0.85 μM and 3.87 μM in BxPc-3 and Panc-1 cells) and enhanced the effects of sorafenib in HCC cells only during hypoxic environments.|
|Brife Description||A protein phosphatase 2A (PP2A) inhibitor(IC50= 0.85 μM and 3.87 μM in BxPc-3 and Panc-1 cells)|
|Related CAS||1026680-07-8 (deleted)|
|Synonyms||(1S,4R)-2-(4-methylpiperazine-1-carbonyl)-7-oxabicyclo[2.2.1]heptane-3-carboxylic acid; LB 100; LB100|
|Solubility||H2O: ≥ 48 mg/mL; DMSO: < 2.9 mg/mL|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||486.9±45.0 ℃ at 760 Torr|
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