|Description||Lavamilast is bio-active molecular as a PDE4 inhibitor but no detailed data has been published yet.|
|Solubility||Soluble in DMSO|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
Eeyarestatin I is a potent inhibitor of endoplasmic reticulum associated protein degradation (ERAD). Eeyarestatin I suppresses ataxin-3 (atx3)-dependent deubiqu...
NAADP tetrasodium salt
NAADP tetrasodium salt is a Ca2+ mobilizing agent. It is an activator of intracellular Ca2+ release via IP3 and cyclic ADP ribose-independent mechanism.
(−)-Epicatechin gallate (ECG) is a natural catechin with a single galloyl group. Like EGCG, it inhibits the growth of cancer cells and has anti-inflammatory eff...
Duloxetine metabolite Para-Naphthol Dulo
Duloxetine metabolite Para-Naphthol Duloxetine is a metabolite of Duloxetine, which is a serotonin-norepinephrine reuptake inhibitor.
Tribromoethanol is a sedative. It is used to anesthetize laboratory animals, particularly rodents, prior to surgery. It has the brand name Avertin as a solution...
Bufotalin is a cardiotoxic bufanolide steroid, cardiac glycoside analogue, secreted by a number of toad species. It is a novel anti-osteoblastoma agent.
PD 130908 is an effective hypoxic cytotoxin as an analogue of RSU 1069, but less potent than the hypoxic cell radiosensitizer RSU 1069. Toxicity toward hypoxic ...
Mebeverine Acid is a metabolite of Mebeverine, an antispasmodic. Mebeverine acid appears to be a valuable marker of oral exposure to Mebeverine.
RD20000, a corticosteroid, is a topical antiinflammatory agent.
(RS)-4-Carboxy-3-hydroxyphenylglycine has been found to be a broad spectrum EAA ligand.
Icaritin was unable to promote proliferation, migration and tube like structure formation by human umbilical vein endothelial cells (HUVECs) in vitro. Icaritin ...
(±)-Vesamicol hydrochloride is an inhibitor of acetylcholine transport (Ki = 2 nM) that blocks the loading of acetylcholine into synaptic vesicles of cholinergi...
GSK 4112, a kind of synthetic agonist of REV-ERBα, could suppress the expression of sorts of genes involved in gluconeogenesis. IC50: 0.4 μM (EC50).
(R)-(-)-PK 11195 is the (R)-enantiomer of PK 11195, which is a peripheral benzodiazepine antagonist with high affinity for PBR in all species. It is used as a d...
Amidantel is a potent anthelminthic agent.
Evans Blue is a potent inhibitor of L-glutamate uptake into synaptic vesicles and is able to antagonize AMPA (IC50=220 nM) and kainate receptor (IC50=150 nM) me...
Amoxapine is a tricyclic dibenzoxazepine (an N-aryl piperazine) which acts similarly to several other tricyclic antidepressants, amoxapine inhibits GLYT2a trans...
Exo1 is a reversible inhibitor of vesicular trafficking between endoplasmic reticulum and Golgi apparatus. Exo1 releases ADP-ribosylation factor (ARF)1 from Gol...
NB-598 is a potent competitive inhibitor of squalene epoxidase (SE).
Diacerin is an inhibitor of pro-inflammatory cytokine Interleukin-1B (IL-1B) production, prescribed for osteoarthritis and chronic inflammatory arthritis.