Lasmiditan - CAS 439239-90-4
Catalog number:
439239-90-4
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H18F3N3O2
Molecular Weight:
377.36
COA:
Inquire
Targets:
5-HT Receptor
Description:
Lasmiditan is a high-affinity, highly selective 5-HT1F receptor agonist(Ki=2.1 nM) for the treatment of acute migraine.
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Purity:
≥98 %
Related CAS:
439239-90-4 (Free base); 613677-28-4 (HCl)
Appearance:
Solid powder
Synonyms:
2,4,6-Trifluoro-N-(6-((1-methylpiperidine-4-yl)carbonyl)pyridin-2-yl)benzamide; COL-144; COL144; COL 144; LY573144; LY-573144; LY 573144; Lasmiditan
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
5-HT1F receptor agonist
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
XEDHVZKDSYZQBF-UHFFFAOYSA-N
InChI:
1S/C19H18F3N3O2/c1-25-7-5-11(6-8-25)18(26)15-3-2-4-16(23-15)24-19(27)17-13(21)9-12(20)10-14(17)22/h2-4,9-11H,5-8H2,1H3,(H,23,24,27)
Canonical SMILES:
O=C(NC1=NC(C(C2CCN(C)CC2)=O)=CC=C1)C3=C(F)C=C(F)C=C3F
Current Developer:
CoLucid Pharmaceuticals
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 439239-90-4 Lasmiditan

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