Laropiprant - CAS 571170-77-9
Catalog number: 571170-77-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H19ClFNO4S
Molecular Weight:
435.91
COA:
Inquire
Targets:
Prostaglandin Receptor
Description:
Laropiprant is a potent, selective DP1 receptor antagonist (Ki=0.57 nM) used in combination with niacin to reduce blood cholesterol (LDL and VLDL).
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Purity:
≥95%
Appearance:
White to off-white solid
Synonyms:
MK-0524; (3R)-4-[(4-chlorophenyl)methyl]-7-fluoro-1,2,3,4-tetrahydro-5-(methylsulfonyl)-cyclopent[b]indole-3-acetic acid 2-[(3R)-4-[(4-chlorophenyl)methyl]-7-fluoro-5-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
A potent, selective DP1 receptor antagonist
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
Melting Point:
173-176 °C
InChIKey:
NXFFJDQHYLNEJK-CYBMUJFWSA-N
InChI:
1S/C21H19ClFNO4S/c1-29(27,28)18-10-15(23)9-17-16-7-4-13(8-19(25)26)20(16)24(21(17)18)11-12-2-5-14(22)6-3-12/h2-3,5-6,9-10,13H,4,7-8,11H2,1H3,(H,25,26)/t13-/m1/s1
Canonical SMILES:
CS(=O)(=O)C1=C2C(=CC(=C1)F)C3=C(N2CC4=CC=C(C=C4)Cl)C(CC3)CC(=O)O
Current Developer:
Merck & Co
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 571170-77-9 Laropiprant

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