|Description||Lanabecestat, also referred to AZD3293,is an orally active and highly permeable potent inhibitor of human β-secretase 1 in clinical development for the treatment of Alzheimer disease with a Ki of 0.4 nM.|
|Brife Description||An oral beta-secretase 1 cleaving enzyme (BACE) inhibitor (Ki= 0.4 nM)|
|Synonyms||(1r,4r)-4-methoxy-5''-methyl-6'-(5-(prop-1-yn-1-yl)pyridin-3-yl)-3'H-dispiro[cyclohexane-1,2'-indene-1',2''-imidazol]-4''-amine; 4-methoxy-5'-methyl-6'-(5-(prop-1-yn-1-yl)pyridin-3-yl)-3'H-dispiro(cyclohexane-1,2'-inden-1',2'-imidazol)-4'-amine; AZD3293|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||621.9±65.0 ℃ at 760 Torr|
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