|Description||Labetalol HCl is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors, used in the treatment of high blood pressure.|
Levalbuterol is a short-acting beta 2 adrenergic agonist. Levalbuterol binds to beta 2 adrenergic receptors and activates intracellular adenyl cyclase to promot...
Octopamine hydrochloride is an α-adrenoceptor agonist.
Lofexidine hydrochloride is the hydrochloride salt form of Lofexidine. Lofexidine, an analogue of clonidine, is an α2A-adrenergic receptor agonist for the treat...
(R)-(-)-Niguldipine Hydrochloride, the less active enantiomer of Niguldipine Hydrochloride, is an L-type calcium channel protein inhibitor and α1A-AR (α1A-adren...
Rec 15/2615 dihydrochloride
Rec 15/2615 dihydrochloride is a selective α1B-adrenoceptor antagonist (Ki= 0.3, 1.9 and 2.6 nM at human α1B, α1A and α1D receptors respectively) potentially fo...
RS 100329 hydrochloride
RS 100329 is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors), with 126- and 50-fold selectivity over human α1B and α1D recept...
Milveterol is a long-acting β(2)-adrenoceptor agonist under the development of GlaxoSmithKline. Phase II trials for the treatment of Chronic obstructive pulmona...
CP-331684 is a β3-adrenergic receptor agonist used as antidiabetic drug.
Alfuzosin HCl is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH).
Methoxamine Hydrochloride is an alpha-1 adrenergic agonist, similar in structure to butaxamine and 2,5-DMA. It causes prolonged peripheral vasoconstriction. It ...
An α1 adrenergic receptor antagonist
DG5128, a new oral hypoglycemic agent, is an orally available preferential antagonist of α2-adrenoceptor with 7.4 times higher affinity toward α2-adrenoceptor t...
Arbutamine is β-adrenergic receptor originated by SICOR. It is a cardiac stimulant. Arbutamine is a synthetic catecholamine with positive chronotropic and inotr...
Vilanterol (GW642444; GW 642444X) is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therap...
Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM, used as a "reliever" inhaler in the management of asthma symptoms and as a...
Landiolol is an ultra-short-acting Beta 1 adrenergic receptor antagonist using for managing supraventricular tachyarrhythmias in sepsis. It is also used as an a...
RS 17053 hydrochloride
RS 17053 is a novel, selective alpha 1A-adrenoceptor antagonist, which displayed high affinity for the alpha 1A-adrenoceptor (pKi and pA2 estimates of 9.1-9.9) ...
CGP-12388 is a beta-adrenoceptor antagonist-derived radioligands. It is used for cardiac PET imaging due to its high hydrophilicity and affinity to beta-adrenoc...
Atipamezole, a 4-substituted imidazole derivative, is an alpha2-adrenoceptor blocker which could be used for animals to recover from the anesthesia by lowering ...
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstru...