|Description||L-NAME is a nonselective inhibitor of nitric oxide synthetases (NOS) for nNOS (bovine), eNOS (human), and iNOS (murine), with Ki of 15 nM, 39 nM and 4.4 μM, respectively.|
|Synonyms||Nω-Nitro-L-arginine methyl ester hydrochloride|
AZ PFKFB3 26
AZ PFKFB3 26 is a selective and potent metabolic kinase PFKFB3 inhibitor with IC50 value of 0.023 μM. It is selective for PFKFB3 over PFKFB1 and PFKFB2 isoforms...
FR 121196 is a potential antidementia drug originated by Fujisawa. Mechanism of Action is not undefined. FR 121196 can ameliorate the impaired memory of rat in ...
GKT137831 attenuates hypoxia-induced H(2)O(2) release, cell proliferation, and TGF-β1 expression and blunted reductions in PPARγ in HPAECs and HPASMCs.
This molecular is a novel non-peptide tachykinin NK3 receptor antagonist and it has a very high affinity for native guinea pig (pK(i) value 7.8) tachykinin NK(3...
PF-1355 is a selective, mechanism-based inhibitor of myeloperoxidase (MPO) (IC50 = 1.5 μM in LPS-stimulated human whole blood) with excellent selectivity for MP...
Ginkgetin is a natural biflavonoid isolated from leaves of Ginkgo biloba L. According to reports, it has anti-inflammatory and anti-cancer effects.
DL-AP4 Sodium salt
The sodium salt form of DL-AP4, which has been found to be a broad spectrum EAA ligand.
Letrozole is a third generation inhibitor of aromatase with IC50 of 0.07-20 nM.