L-778123 HCl - CAS 253863-00-2
Catalog number: B0084-176694
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H20ClN5O
Molecular Weight:
405.88
COA:
Inquire
Targets:
Farnesyl Transferase
Description:
L-778123 is an inhibitor of FPTase and GGPTase-I, which was developed in part because it can completely inhibit Ki-Ras prenylation.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-176694 50 mg $398 In stock
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Purity:
98%
Related CAS:
183499-57-2 (Free base)
Appearance:
white solid powder
Synonyms:
4-((5-((4-(3-chlorophenyl)-3-oxopiperazin-1-yl)methyl)-1H-imidazol-1-yl)methyl)benzonitrile hydrochloride; L778123; L-778123; L 778123; L778,123; L-778,123; L 778,123 HCl
Solubility:
Soluble in DMSO, not in water
Storage:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
MSDS:
Inquire
Shelf Life:
2 years if stored properly
InChIKey:
YNBSQYGTJLIPJS-UHFFFAOYSA-N
InChI:
1S/C22H20ClN5O.ClH/c23-19-2-1-3-20(10-19)28-9-8-26(15-22(28)29)14-21-12-25-16-27(21)13-18-6-4-17(11-24)5-7-18;/h1-7,10,12,16H,8-9,13-15H2;1H
Canonical SMILES:
N#CC1=CC=C(CN2C(CN3CC(N(C4=CC=CC(Cl)=C4)CC3)=O)=CN=C2)C=C1.[H]Cl
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