KY1220 - CAS 292168-79-7
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C14H10N4O3S
Molecular Weight:
314.32
COA:
Inquire
Targets:
Wnt | β-catenin
Description:
KY1220 is a novel inhibitor of the Wnt/ß-catenin pathway, destabilizing both β-catenin and Ras via targeting the Wnt/β-catenin pathway (IC50= 2.1 μM in HEK293 reporter cells).
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Synonyms:
(5Z)-5-[[1-(4-nitrophenyl)pyrrol-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Solubility:
DMSO: ≥100 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Density:
1.54±0.1 g/cm3
InChIKey:
FMLUAKSJMUPACD-WQLSENKSSA-N
InChI:
1S/C14H10N4O3S/c19-13-12(15-14(22)16-13)8-11-2-1-7-17(11)9-3-5-10(6-4-9)18(20)21/h1-8H,(H2,15,16,19,22)/b12-8-
Canonical SMILES:
C1=CN(C(=C1)C=C2C(=O)NC(=S)N2)C3=CC=C(C=C3)[N+](=O)[O-]
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Chemical Structure

CAS 292168-79-7 KY1220

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