|Description||KT 5823 is a cell-permeable, selective inhibitor of cGMP-dependent protein kinase (PKG) (Ki values are 0.23, 4 and > 10 μM for inhibition of PKG, PKC and PKA respectively). KT 5823 is often used in intact cells to assess the role of PKG in signaling, , although there are cases where it poorly inhibits PKG in cells.|
|Synonyms||2,3,9,10,11,12-hexahydro-10R-methoxy-2,9-dimethyl-1-oxo-9S,12R-epoxy-1H-diindolo[1,2,3-fg:3’,2’,1’-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid, methyl ester;|
|Solubility||Soluble to 50 mM in DMSO|
|Storage||Desiccate at -20°C|
|Boiling Point||629.2±55.0 °C | Condition: Press: 760 Torr|
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