|Description||Kevetrin hydrochloride is a water-soluble small molecule with potential antineoplastic activity.|
|Synonyms||UNII-NL6L2371DP; thioureidobutyronitrile; 3-cyanopropyl carbamimidothioate;hydrochloride; Carbamimidothioic acid, 3-cyanopropyl ester, monohydrochloride|
|Solubility||Soluble in DMSO|
|Storage||Store at -20 °C|
|Application||Inhibiting cancer cell growth and causing tumor cell apoptosis.|
|Quality Standard||Enterprise Standard|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly|
RO5045337, also known as R7112, RG7112, is a MDM2 antagonist with potential antineoplastic activity. RO5045337 binds to MDM2, thereby preventing the binding of...
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RITA (NSC 652287)
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Kevetrin hydrochloride is a water-soluble small molecule with potential antineoplastic activity.
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MI-773 (SAR405838) is an orally available MDM2 antagonist with Ki of 0.88 nM. Phase 1.