KDM5-inhibitor
Catalog number: B0084-284866
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C16H14N4O
Molecular Weight:
278.315
COA:
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Targets:
Histone Demethylase
Description:
KDM5-inhibitor is an analog of CPI-455, a selective KDM5 inhibitor. CPI-455 increases levels of H3K4 trimethylation (H3K4me3) and decreases the number of DTPs in multiple cancer cell lines treated with standard chemotherapy or targeted agents. It reduces survival of drug-tolerant cancer cells.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-284866 10 mg $198 In stock
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Synonyms:
7-oxo-5-phenyl-6-propyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile
MSDS:
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InChIKey:
GDYICSDRFQBRDX-UHFFFAOYSA-N
InChI:
InChI=1S/C16H14N4O/c1-2-6-13-14(11-7-4-3-5-8-11)19-15-12(9-17)10-18-20(15)16(13)21/h3-5,7-8,10,18H,2,6H2,1H3
Canonical SMILES:
CCCC1=C(N=C2C(=CNN2C1=O)C#N)C3=CC=CC=C3
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