|Description||JZP 361 is a reversible, potent and selective inhibitor of human recombinant MAGL (hMAGL) with IC50 value of 46 nM. It shows affinity for H1 receptors but shows no activity at cannabinoid receptors. It has MAGL-inhibitory and antihistaminergic and may be a novel dual-acting pharmacological tool.|
|Purity||≥99% by HPLC|
|Synonyms||JZP-361; JZP 361; JZP361; [4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4-triazol-1-yl)methanone|
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JZP 361 is a reversible, potent and selective inhibitor of human recombinant MAGL (hMAGL) with IC50 value of 46 nM. It shows affinity for H1 receptors but shows...
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