JNJ-26146900 - CAS 868691-50-3
Catalog number: 868691-50-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C15H15F3N2O3S
Molecular Weight:
360.35
COA:
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Targets:
Androgen Receptor
Description:
JNJ-26146900 is a selective, nonsteroidal androgen receptor modulator with tissue-selective activity in rats. It can bind to the rat AR with a Ki of 400nM and act as a pure androgen antagonist in an in vitro cell-based assay. But no development was reported for the treatment of Bone disorders and Cancer till now.
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Purity:
98%
Appearance:
Powder
Synonyms:
(-)(R)-2-(2-Ethylsulfonyl-1-hydroxy-1-methylethyl)-6-trifluoromethyl-1H-indole-5-carbonitrile
Solubility:
Soluble in DMSO
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Bone disorders; Cancer
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
UJGGNFGSHPHGNE-AWEZNQCLSA-N
InChI:
1S/C15H15F3N2O3S/c1-3-24(22,23)8-14(2,21)13-5-9-4-10(7-19)11(15(16,17)18)6-12(9)20-13/h4-6,20-21H,3,8H2,1-2H3/t14-/m0/s1
Canonical SMILES:
CCS(=O)(=O)C[C@@](C)(c1cc2cc(c(cc2[nH]1)C(F)(F)F)C#N)O
Current Developer:
Janssen Research & Development
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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