Ipatasertib - CAS 1001264-89-6
Catalog number:
1001264-89-6
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
COA:
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Targets:
Akt
Description:
Ipatasertib, also known as GDC-0068 is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity. Akt inhibitor GDC-0068 binds to and inhibits the activity of Akt in a non-ATP-competitive manner, which may result in the inhibition of the PI3K/Akt signaling pathway and tumor cell proliferation and the induction of tumor cell apoptosis. Activation of the PI3K/Akt signaling pathway is frequently associated with tumorigenesis and dysregulated PI3K/Akt signaling may contribute to tumor resistance to a variety of antineoplastic agents.
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Appearance:
Solid powder
Synonyms:
GDC-0068; GDC0068; GDC 0068; RG7440; RG-7440; RG 7440; Ipatasertib
MSDS:
Inquire
Current Developer:
Genentech/Array BioPharma Inc.
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CAS 1001264-89-6 Ipatasertib

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