|Description||Iopamidol is a nonionic, low-osmolar iodinated contrast agent, developed by Bracco.|
|Synonyms||Iopamiro; Isovue; Iopamiron; Niopam|
KPU-300, a diketopiperazine derivative, has been found to be an antimicrotubule agent and exhibit cytotoxicity against HT-29 cells. IC50: 7.0 nM.
Lotilaner is an insecticide and veterinary drug.
LUF 6283 is a partial hydroxycarboxylic acid receptor 2 agonist. It can effectively lower plasma lipid levels.
Gimeracil is a pyridine derivative with antitumor activity. Gimeracil enhances the antitumor activity of fluoropyrimidines by competitively and reversibly inhib...
Cinobufagin can inhibit the proliferation of U-2OS cells, and induce cell apoptosis. The potential mechanism of Cinobufagin-induced apoptosis may be related to ...
Pseudobufarenogin is a natural compound extracted from toad species with unknown details.
BVT 948 is a non-competitive and cell-permeable inhibitor of protein tyrosine phosphatases (PTPs) (IC50 = 0.09 - 1.7 μM). BVT 948 displays irreversible inhibiti...
FR-900490 is a new type of immunoactive substance isolated from Disocia sp. F-11809. It is effective in reversing the damage to bone marrow caused by mitomycin ...
GYKI-20238 is a thiazolidine compound with anti-amnesic activity.
ARV-825, a BRD4 inhibitor, has extensive anti-AML activity and modulates tumor microenvironment and metabolism to overcome stromamediated drug resistance. DC50...
A 438079 hydrochloride
A 438079 hydrochloride is a competitive P2X7 receptor antagonist with pIC50 value of 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell li...
Azacyclonol, also known as γ-pipradol, is a drug used to diminish hallucinations in psychotic individuals.
OT-R antagonist 1
OT-R antagonist 1 is a nonpeptide OT-R antagonist, inhibitis IP3-Synthesis, rat OT-R (IC50 = 8 nM).
MDL 12330A hydrochloride
MDL 12330A is an adenylyl cyclase inhibitor. It can also inhibit cAMP and cGMP phosphodiesterases, and block slow extracellular and store-operated Ca2+ entry in...
BI-44847 is a synthetic bio-active chemical had been in phase II clinical trials for the treatment of type 2 diabetes.
A12B4C3 is a potent and selective inhibitor of polynucleotide kinase/phosphatase (PNKP) (IC50 = 60 nM), a DNA repair enzyme. A12B4C3 is inactive to calcineurin,...
GLPG 0974 is a potent FFA2 antagonist (IC50 = 9 nM) with selectivity for FFA2 over FFA3. It was shown that GLPG 0974 inhibited acetate-induced human neutrophil ...
Xenopsin, the neurotensin-like octapeptide fromXenopusskin at the carboxyl terminus of its precursor, shows sequence homology to mammalian neurotensin and share...
Aminohippurate Sodium is a diagnostic agent that is used to help differentiate and characterized organic anion transporter (OAT) isoforms. It is useful in medic...
ABT 089 dihydrochloride
ABT 089 dihydrochloride is a selective α4β2 nicotinic acetylcholine receptor partial agonist (Ki = 16 nM) with >1000-fold and >10,000-fold selectivity for α4β2 ...